Philip V Felice

US Patent:

8304404, Nov 6, 2012

Filed:

Apr 5, 2012

Appl. No.:

13/440693

Inventors:

Harry G. Brittain - Milford NJ, US
Philip V. Felice - Smithtown NY, US

Assignee:

Theaprin Pharmaceuticals Inc. - Hauppauge NY

International Classification:

A61K 31/60
A61K 31/12

US Classification:

514165, 514676

Abstract:

An aspirin-theanine cocrystal composition including a quantity of acetylsalicylic acid and a quantity of a theanine enantiomer combined with the quantity of acetylsalicylic acid in a mixture. The theanine enantiomer may be L-theanine, D-theanine, or DL-theanine.

US Patent:

8476250, Jul 2, 2013

Filed:

Jan 2, 2013

Appl. No.:

13/732807

Inventors:

Philip V. Felice - Smithtown NY, US

Assignee:

Theaprin Pharmaceuticals Inc. - Hauppauge NY

International Classification:

A61K 31/60
A61K 31/12

US Classification:

514165, 514676

Abstract:

A method of treatment using a water-soluble cocrystal composition contains a quantity of acetylsalicylic acid and a quantity of a theanine enantiomer selected from an alpha variant of theanine or a beta variant of theanine or other form of theanine.

US Patent:

20100286099, Nov 11, 2010

Filed:

May 8, 2009

Appl. No.:

12/437735

Inventors:

Harry G. Brittain - Milford NJ, US
Philip V. Felice - Smithtown NY, US

International Classification:

A61K 31/60
A61P 35/00

US Classification:

514162

Abstract:

A water-soluble aspirin-theanine cocrystal composition which includes a quantity of acetylsalicylic acid and a quantity of a theanine enantiomer associated with the quantity of acetylsalicylic acid. The composition may be created by a method including the steps of: (i) providing a quantity of acetylsalicylic acid; (ii) adding a quantity of a theanine enantiomer to the quantity of acetylsalicylic acid to form a mixture comprising the quantity of acetylsalicylic acid and the enantiomer of theanine; (iii) wetting the mixture; and (iv) grinding the mixture for a length of time sufficient to produce a dried crystalline mass. The water-soluble cocrystal composition is suitable for intravenous administration, preferably to humans.

US Patent:

20130012482, Jan 10, 2013

Filed:

Sep 14, 2012

Appl. No.:

13/617508

Inventors:

Harry G. Brittain - Milford NJ, US
Philip V. Felice - Smithtown NY, US

Assignee:

THEAPRIN PHARMACEUTICALS INC. - Hauppauge NY

International Classification:

A61K 31/616
A61P 29/00

US Classification:

514162

Abstract:

A water-soluble cocrystal composition contains a quantity of acetylsalicylic acid and a quantity of a theanine enantiomer selected from an alpha variant of theanine or a beta variant of theanine or other form of theanine.

US Patent:

20130345183, Dec 26, 2013

Filed:

Aug 14, 2013

Appl. No.:

13/967027

Inventors:

Philip V. Felice - Smithtown NY, US

Assignee:

THEAPRIN PHARMACEUTICALS INC. - Hauppauge NY

International Classification:

A61K 31/616
A61K 31/198

US Classification:

514162

Abstract:

A method of treating rheumatoid arthritis using a water-soluble cocrystal composition contains a quantity of acetylsalicylic acid and a quantity of a theanine enantiomer selected from an alpha variant of theanine or a beta variant of theanine or other form of theanine.

US Patent:

20170143648, May 25, 2017

Filed:

Nov 17, 2016

Appl. No.:

15/353989

Inventors:

- Hauppauge NY, US
Philip V. Felice - Smithtown NY, US

Assignee:

THEAPRIN PHARMACEUTICALS INC. - Hauppauge NY

International Classification:

A61K 31/138
A61K 9/00

Abstract:

Methods of treating and preventing conditions by employing cocrystal compositions of metoprolol and dabigatran bases with enantiomers of theanine.

US Patent:

20170143838, May 25, 2017

Filed:

Oct 3, 2016

Appl. No.:

15/284074

Inventors:

- Hauppauge NY, US
Philip V. Felice - Smithtown NY, US

Assignee:

THEAPRIN PHARMACEUTICALS INC. - Hauppauge NY

International Classification:

A61K 47/48
A61K 31/138
A61K 31/4439
A61K 31/198

Abstract:

Cocrystal compositions of metoprolol and dabigatran bases with enantiomers of theanine.

US Patent:

20170144964, May 25, 2017

Filed:

Nov 17, 2016

Appl. No.:

15/353927

Inventors:

- Hauppauge NY, US
Philip V. Felice - Smithtown NY, US

Assignee:

THEAPRIN PHARMACEUTICALS INC. - Hauppauge NY

International Classification:

C07C 237/08
C07D 401/12
C07C 217/54

Abstract:

Methods of making cocrystal compositions of metoprolol and dabigatran bases with enantiomers of theanine.